| 英文名稱 | Pristimerin (Synonyms: Celastrol methyl ester) |
|---|---|
| 中文名稱 | 扁蒴藤素 |
| CAS號 | 1258-84-0 |
| 分子式 | C30H40O4 |
| 分子量 | 464.64 |
| 外觀 | Orange to reddish brown powder |
| 儲存條件 | Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years). |
| 英文名稱 | Pristimerin (Synonyms: Celastrol methyl ester) |
|---|---|
| 中文名稱 | 扁蒴藤素 |
| CAS號 | 1258-84-0 |
| 分子式 | C30H40O4 |
| 分子量 | 464.64 |
| 外觀 | Orange to reddish brown powder |
| 儲存條件 | Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years). |
Pristimerin is a triterpenoid and an antitumor agent. Induces caspase-dependent apoptosis by inhibiting the chymotrypsin-like activity of the proteasome.
Discovery of potent and reversible monoacylglycerol lipase inhibitors.
PMID: 19875078 PMCID: PMC3034734 DOI: 10.1016/j.chembiol.2009.09.012
PMID: 26548348 DOI: 10.1016/j.intimp.2015.11.001